Our Science

OUR SCIENCE

Congress Presentations

This section includes posters and presentations related to Arvinas’ PROTAC science, discovery compounds, and clinical-stage assets presented at scientific congresses in the past three years.


ESMO 2023 | Madrid, Spain

Oct 20 - 24, 2023

Poster
Vepdegestrant, a PROteolysis TArgeting Chimera (PROTAC) Estrogen Receptor Degrader, in Estrogen Receptor+/Human Epidermal Growth Factor Receptor 2-Advanced Breast Cancer: Update of Dose Escalation Results From a Phase 1/2 Trial

EP Hamilton et al.

ESMO 2023 | Madrid, Spain

Oct 20 - 24, 2023

Poster
Phase 1/2 Study of Bavdegalutamide, a PROteolysis TArgeting Chimera (PROTAC) Androgen Receptor Degrader, in Metastatic Castration-Resistant Prostate Cancer: Radiographic Progression-Free Survival in Patients With Androgen Receptor Ligand-Binding Domain Mutation

DP Petrylak et al.

ISSX 2023 | Boston, MA

Sep 10 - 13, 2023

Poster
In Vitro Evaluation of PROTAC® Androgen Receptor Degrader ARV-766 for Cytochrome P450- and Transporter-Mediated Drug-Drug Interaction

JG Zhang et al.

ACCP 2023 | Bellevue, WA

Sep 10 - 12, 2023

Poster
Drug-Drug Interaction Study of the PROteolysis TArgeting Chimera (PROTAC) Androgen Receptor Degrader Bavdegalutamide in Combination With the CYP3A4 Inhibitor Itraconazole in Healthy Volunteers

J Alicea et al.

ACCP 2023 | Bellevue, WA

Sep 10 - 12, 2023

Poster
The Effect of Food and the Proton Pump Inhibitor Esomeprazole on the Single-Dose Pharmacokinetics and Safety of the PROteolysis Targeting Chimera (PROTAC) Androgen Receptor Degrader Bavdegalutamide in Healthy Volunteers

J Alicea et al.

ACCP 2023 | Bellevue, WA

Sep 10 - 12, 2023

Poster
The Effect of Food and the Proton Pump Inhibitor Esomeprazole on the Single-Dose Pharmacokinetics and Safety of ARV-766, a PROteolysis TArgeting Chimera (PROTAC) Androgen Receptor Degrader, in Healthy Volunteers

J Alicea et al.

MDS 2023 | Copenhagen, Denmark

Aug 27 - 31, 2023

Poster
Development of Potent, Orally Bioavailable, and Highly Selective LRRK2 PROTAC® Degrader Molecules as Potential Disease Modifying Therapeutics for Parkinson’s Disease

K Kelly et al.

MDS 2023 | Copenhagen, Denmark

Aug 27 - 31, 2023

Poster
LRRK2 PROTAC® Degrader Molecules Induce Robust Biomarker Responses in Preclinical In Vivo Pharmacology Studies Following Acute and Chronic Oral Dosing

J Meredith Jr. et al.

ASCO 2023 | Chicago, IL

Jun 2 - 6, 2023

Poster
TACTIVE-U: Phase 1b/2 Umbrella Study of ARV-471, a PROteolysis TArgeting Chimera (PROTAC) Estrogen Receptor (ER) Degrader, Combined with Other Anticancer Treatments in ER+ Advanced or Metastatic Breast Cancer

RM Layman et al.